Listar QUIO_Articles por autoría "c5931120-4d21-4985-bc69-534538e0bdf3"
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Aryl urea based scaffolds for multitarget drug discovery in anticancer immunotherapies
Martín Beltrán, Celia; Gil-Edo, Raquel; Hernández Ribelles, Germán; Agut, Raúl; Marí Mezquita, Pilar; Carda, Miguel; Falomir, Eva MDPI (2021-04-06)Twenty-one styryl and phenethyl aryl ureas have been synthetized and biologically evaluated as multitarget inhibitors of Vascular endothelial growth factor receptor-2 VEGFR-2 and programmed death-ligand-1 (PD-L1) proteins ... -
Exploring BenzylethoxyAryl Urea Scaffolds for Multitarget Immunomodulation Therapies
Gil-Edo, Raquel; Hernández Ribelles, Germán; Royo, Santiago; Thawait, Natasha; Serrels, Alan; Carda, Miguel; Falomir, Eva MDPI (2023-05-11)Thirteen benzylethoxyaryl ureas have been synthesized and biologically evaluated as multitarget inhibitors of VEGFR-2 and PD-L1 proteins to overcome resistance phenomena offered by cancer. The antiproliferative activity ...