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Design, synthesis and antimalarial evaluation of novel thiazole derivatives
Bueno, José María; Carda, Miguel; Crespo, Benigno; Cuñat, Ana Carmen; De Cozar, Cristina; León, María Luisa; Marco, J. Alberto; Roda, Nuria; Sanz-Cervera, Juan F. Elsevier (2016)As part of our medicinal chemistry program’s ongoing search for compounds with antimalarial activity, we prepared a series of thiazole analogs and conducted a SAR study analyzing their in vitro activities against the ...