2024-03-28T08:49:31Zhttps://repositori.uji.es/oai/requestoai:repositori.uji.es:10234/1664522022-10-28T13:12:19Zcom_10234_116245com_10234_158177com_10234_10col_10234_166357
00925njm 22002777a 4500
dc
Moreno-Rius, Josep
author
Pubill Sánchez, David
author
Escubedo Rafa, Elena
author
Camarasa Garcia, Jordi
author
MIQUEL, MARTA
author
2017
Introducción: La 3,4-Methylenedioxypyrovalerone (mdpv) es un componente de las
denominadas sales de baño, aparecidas en el mercado a final de la década del 2000
debido a la falta de precursores de síntesis de mdma, y su uso va en aumento. El ob-
jetivo de este trabajo es clarificar sus características farmacológicas y potencialidades
adictivas. Método: Mediante búsquedas en PubMed, 21 estudios relacionados con la
química, farmacología o potencial adictivo del mdpv fueron seleccionados. Resulta-
dos: El mdpv muestra ser capaz de inducir una potente hiperlocomoción, preferencias
condicionadas, sensibilización conductual, autoadministración y altos puntos de corte
en pruebas de razón progresiva. Conclusión: Los estudios revisados apuntan a que
el mdpv es un potente psicoestimulante con un potencial adictivo similar al de la cocaí-
na o la metanfetamina. Su abuso continuado podría llevar a una epidemia de adictos
al mdpv.
Introduction: 3,4-Methylenedioxypyrovalerone (mdpv) is a major component of the new
psychoactive substances termed “bath salts”. These substances appeared on the drug
market at the end of the last century given the lack of mdma precursors, caused by its
worldwide prosecution by governments and police agencies, and its growing use. The
goal of this work was to clarify its pharmacological features and addiction-like potentiali-
ties. Methods: By PubMed searches, 21 studies related to mdpv chemistry, pharmaco
logy or addictive features were selected. Results: mdpv is seen to be able to induce
potent hyperlocomotion, conditioned place preference, behavioural sensitisation, self-
administration and high breakpoints in progressive ratio schedules. Conclusion: The
reviewed studies indicate that mdpv is a powerful psychostimulant with a similar addictive
potential to that of cocaine or methamphetamine. Its abuse can lead to an epidemic of
mdpv addicts.
2443-9827
http://hdl.handle.net/10234/166452
http://dx.doi.org/10.6035/AgoraSalut.2017.4.25
progressive ratio
hyperlocomotion
self-administration
conditioned preference
bath salts
mdpv
sales de baño
preferencia condicionada
autoadministración
razón progresiva
Locomotor activating effects and addiction-like features of MDPV as assessed in preclinical studies: a review.